Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
| more potent alpha 1 than alpha 2 agonist |
|
|
Term
|
Definition
|
|
Term
| all alpha 2 receptors inhibit _______ by g proein interaction causing ______ |
|
Definition
| adenyl cyclase; hyperpolarization |
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
| more alpha than beta agonist |
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
| more beta 2 than isoproterenol but less than albuterol agonist |
|
|
Term
|
Definition
|
|
Term
|
Definition
| relatively selective beta 2 agonist |
|
|
Term
|
Definition
| beta 2 agonist- more than albuterol |
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
| forms alpha-methyl NE-- acts as a false transmitter-- less potent that NE |
|
|
Term
|
Definition
| inhibits amine re-uptake pump, thus causing increased stimulation (indirect effect) agonist |
|
|
Term
|
Definition
| mixed- direct/ indirect agonist |
|
|
Term
|
Definition
| mixed agonist- both alpha and beta |
|
|
Term
|
Definition
| potent sympathomimetic- direct alpha 1, beta 1, beta 2 activity in addition to triggering the release of catacholamines from the nerve terminal (mixed effects) |
|
|
Term
|
Definition
| indirect adrenergic agonist |
|
|
Term
|
Definition
| alpha1 and alpha 2 antagonist- irreversible covalent bonding |
|
|
Term
|
Definition
| alpha 1 and alpha 2 competitive antagonist |
|
|
Term
|
Definition
| selective alpha 1 antagonist |
|
|
Term
|
Definition
| selective alpha 1 antagonist-- less potent than prazosin |
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
| slective alpha 1a antagonist |
|
|
Term
|
Definition
| competitive alpha 2 antagonist |
|
|
Term
|
Definition
| prototype beta antagonist |
|
|
Term
|
Definition
| non selective beta antagonist |
|
|
Term
|
Definition
| non selective beta antagonist |
|
|
Term
|
Definition
| non selective bea antagonist with some sympahetic agonist activity |
|
|
Term
|
Definition
| alpha 1, beta 1 &2 antagonist |
|
|
Term
|
Definition
| alpha 1, beta 1& 2 atnagonist |
|
|
Term
|
Definition
| beta 1 antagonist but also partial sympathetic agonist (non-selective) |
|
|
Term
|
Definition
|
|
Term
|
Definition
|
|
Term
|
Definition
| inhibitor of tyrosine hydrozylase |
|
|
Term
|
Definition
| taken up into adrenergic nerve terminal and destroys the cell |
|
|
Term
|
Definition
| blocks catecholamine release from nerve terminal |
|
|
Term
|
Definition
| inhibits storage of catecholamines and serotonin in granules leading to depletion |
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|
